Top Picks: new discover of 22468-26-4

Here is just a brief introduction to this compound(22468-26-4)Product Details of 22468-26-4, more information about the compound(4-Hydroxypicolinic acid) is in the article, you can click the link below.

In general, if the atoms that make up the ring contain heteroatoms, such rings become heterocycles, and organic compounds containing heterocycles are called heterocyclic compounds. An article called 4-(Tetrazolylalkyl)piperidine-2-carboxylic acids. Potent and selective N-methyl-D-aspartic acid receptor antagonists with a short duration of action, published in 1991-01-31, which mentions a compound: 22468-26-4, Name is 4-Hydroxypicolinic acid, Molecular C6H5NO3, Product Details of 22468-26-4.

A series of trans- and cis-4-(tetrazolylalkyl)piperidine-2-carboxylic acids I (R = H, Me) and II (n = 1, R = H, Me; n = 2-4, R = H) as potent and selective N-methyl-D-aspartic acid (NMDA) receptor antagonists were prepared and evaluated in vitro in both receptor binding assays and in a cortical-wedge preparation to determine affinity, potency, and selectivity. The new amino acids were also evaluated in vivo for their ability to block NMDA-induced convulsions in neonatal rats and NMDA-induced lethality in mice. The most potent compound of this series was I (R = H). I (R = H) blocked both NMDA-induced convulsions in neonatal rats and NMDA-induced lethality in mice. This is the first example of an NMDA receptor antagonist that incorporates a tetrazole moiety as an ω-acid bioisostere. These amino acid antagonists are also unique from their phosphonic acid counterparts in that they have a shorter duration of action in vivo.

Here is just a brief introduction to this compound(22468-26-4)Product Details of 22468-26-4, more information about the compound(4-Hydroxypicolinic acid) is in the article, you can click the link below.

Reference:
Chiral Catalysts,
Chiral catalysts – SlideShare